English Journal
- Comparative Evaluation of Opioid-Induced Changes in Immune Reactivity of CBA Mice.
- Cheido MA1, Gevorgyan MM, Zhukova EN.
- Bulletin of experimental biology and medicine.Bull Exp Biol Med.2014 Jan;156(3):363-5. doi: 10.1007/s10517-014-2349-8. Epub 2014 Jan 16.
- Comparison of IgM and IgG-humoral immune response of CBA mice immunized with SE (5 × 10(8) cells) to activation of μ- (DAGO, 100 μg/kg) and δ2- (DSLET, 100 μg/kg) opioid receptors was studied. Different effects of opioids on IgM and IgG antibody production and peripheral blood and spleen
- PMID 24771376
- N-terminal guanidinylation of TIPP (Tyr-Tic-Phe-Phe) peptides results in major changes of the opioid activity profile.
- Weltrowska G1, Nguyen TM, Chung NN, Wilkes BC, Schiller PW.
- Bioorganic & medicinal chemistry letters.Bioorg Med Chem Lett.2013 Sep 15;23(18):5082-5. doi: 10.1016/j.bmcl.2013.07.036. Epub 2013 Jul 23.
- Derivatives of peptides of the TIPP (Tyr-Tic-Phe-Phe; Tic=1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid) family containing a guanidino (Guan) function in place of the N-terminal amino group were synthesized in an effort to improve their blood-brain barrier permeability. Unexpectedly, N-terminal a
- PMID 23932788
Japanese Journal
- Introduction of F_3-Threonine to the Hexapeptide, DSLET : Investigation of the Effect of Fluorine Atoms toward Peptidic Conformations
- Introduction of F3-Threonine to the Hexapeptide, DSLET: Investigation of the Effect of Fluorine Atoms toward Peptidic Conformations
Related Links
- How is D-Ser2-Leu-Enkephalin-Thr6 (opioid) abbreviated? DSLET stands for D-Ser2-Leu-Enkephalin-Thr6 (opioid). DSLET is defined as D-Ser2-Leu-Enkephalin-Thr6 (opioid) very rarely. Printer friendly Menu Search New search NFL, ...
- Leu-Enkephalin-Thr [D-Ser2] / Delta-Receptor Peptide / DSLET 販売元 和光純薬工業(株) 販売元コード 301-37013 製造元 Anygen Co., Ltd. 製造元コード AGP-8610 CAS.NO 分子式 分子量 保存条件 冷凍 (ドライアイス輸送) 適用法規 ...
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★リンクテーブル★
[★]
- 英
- opioid
- 同
- 類麻薬
- 関
- オピオイド受容体
作用
縮瞳
- モルフィンと多くのμ,κアゴニストは瞳孔の縮小を引き起こす。これは瞳孔を支配する副交感神経の興奮による。μアゴニストを中毒量投与すると縮瞳し、pinpoints pupupilsはpathognomonicである。(GOO.559)
オピオイドとオピオイド類似物質の作用
- GOO.552
+アゴニスト ーアンタゴニスト P partial agonist
各鎮痛薬のオピオイド受容体への作用
- μ受容体 κ受容体
- レミフェンタニル +++ ー
- フェンタニル +++ -
- モルヒネ +++ +
- ペチジン ++ +
- トラマドール + -
- ペンタゾシン ー ++
- ブプレノルフィン P ー
- ナロキソン ー -