β-フナルトレキサミン
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Japanese Journal
- ドコサヘキサエン酸による抗侵害作用の発現機序の解明
- 西中 崇,松本 健吾,中本 賀寿夫 [他],安保 明博,万倉 三正,小山 豊,徳山 尚吾
- YAKUGAKU ZASSHI 133(5), 493-499, 2013
- … This effect was abolished by pretreated with the β-funaltrexamine (β-FNA), a μ-opioid receptor antagonist, and the nartrindole (NTI), a δ-opioid receptor antagonist, but not by the nor-binaltorphimine (nor-BNI), a κ-opioid receptor antagonist. … Furthermore, the pretreatment of anti β-endorphin antiserum inhibited DHA-induced antinociception. … The plasma levels of β-endorphin increased 30 min after DHA administration. …
- NAID 130003361941
- Effects of Loperamide on Mechanical Allodynia Induced by Herpes Simplex Virus Type-1 in Mice
- Sasaki Atsushi,Nakashima Yasutaka,Takasaki Ichiro [他],ANDOH Tsugunobu,SHIRAKI Kimiyasu,KURAISHI Yasushi
- Journal of pharmacological sciences 104(3), 218-224, 2007-07-20
- … The peripheral opioid receptor antagonist naloxone methiodide (0.1 mg/kg, s.c.) and the μ-opioid receptor-selective antagonist β-funaltrexamine (40 nmol/site, intraplantar and 20 mg /kg, s.c.) antagonized the anti-allodynic effects of systemic and local loperamide. …
- NAID 10024314645
- Antinociceptive Effect of Shakuyakukanzoto, a Kampo Medicine, in Diabetic Mice
- Omiya Yuji,Suzuki Yasuyuki,Yuzurihara Mitsutoshi [他],MURATA Mikio,ABURADA Masaki,KASE Yoshio,TAKEDA Shuichi
- Journal of pharmacological sciences 99(4), 373-380, 2005-12-20
- … The antinociceptive activity of shakuyakukanzoto in diabetic mice was not antagonized by β-funaltrexamine, naltrindole, or nor-binaltorphimine. …
- NAID 10025731766
Related Links
- Sigma-Aldrich offers Sigma-O003, β-Funaltrexamine hydrochloride for your research needs. Find product specific information including CAS, MSDS, protocols and references.
- 1 May 2007 ... Interestingly, neither the nonselective opioid receptor antagonist, naltrexone nor β-funaltrexamine (β-FNA), a highly selective MOR antagonist, blocked fentanyl mediated inhibition of TNFα induced CXCL10 expression. Rather ...
Related Pictures
★リンクテーブル★
[★]
- 英
- opioid
- 同
- 類麻薬
- 関
- オピオイド受容体
作用
縮瞳
- モルフィンと多くのμ,κアゴニストは瞳孔の縮小を引き起こす。これは瞳孔を支配する副交感神経の興奮による。μアゴニストを中毒量投与すると縮瞳し、pinpoints pupupilsはpathognomonicである。(GOO.559)
オピオイドとオピオイド類似物質の作用
- GOO.552
+アゴニスト ーアンタゴニスト P partial agonist
各鎮痛薬のオピオイド受容体への作用
- μ受容体 κ受容体
- レミフェンタニル +++ ー
- フェンタニル +++ -
- モルヒネ +++ +
- ペチジン ++ +
- トラマドール + -
- ペンタゾシン ー ++
- ブプレノルフィン P ー
- ナロキソン ー -