- 関
- GABAergic
WordNet
- supply with a gate; "The house was gated"
- restrict (school boys'
- total admission receipts at a sports event
- a computer circuit with several inputs but only one output that can be activated by particular combinations of inputs (同)logic gate
- a movable barrier in a fence or wall
- passageway (as in an air terminal) where passengers can embark or disembark
- control with a valve or other device that functions like a gate
- a gangsters pistol (同)rod
PrepTutorEJDIC
- (…への)『門』,通用門《+『to』(『of』)+『名』》;(門の)とびら / (ダム・運河などの)水門 / (競技場・劇場などの)[有料]入場者数 / (またgate money)総入場料
- ピストル,はじき
- General Admiral / (またGa)Georgia
UpToDate Contents
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English Journal
- Discovery of sarolaner: A novel, orally administered, broad-spectrum, isoxazoline ectoparasiticide for dogs.
- McTier TL1, Chubb N2, Curtis MP2, Hedges L2, Inskeep GA2, Knauer CS2, Menon S2, Mills B2, Pullins A2, Zinser E2, Woods DJ2, Meeus P2.
- Veterinary parasitology.Vet Parasitol.2016 May 30;222:3-11. doi: 10.1016/j.vetpar.2016.02.019. Epub 2016 Feb 23.
- The novel isoxazoline ectoparasiticide, sarolaner, was identified during a lead optimization program for an orally-active compound with efficacy against fleas and ticks on dogs. The aim of the discovery program was to identify a novel isoxazoline specifically for use in companion animals, beginning
- PMID 26961590
- Emamectin is a non-selective allosteric activator of nicotinic acetylcholine receptors and GABAA/C receptors.
- Xu X1, Sepich C2, Lukas RJ3, Zhu G4, Chang Y5.
- Biochemical and biophysical research communications.Biochem Biophys Res Commun.2016 May 13;473(4):795-800. doi: 10.1016/j.bbrc.2016.03.097. Epub 2016 Apr 2.
- Avermectins are a group of compounds isolated from a soil-dwelling bacterium. They have been widely used as parasiticides and insecticides, acting by relatively irreversible activation of invertebrate chloride channels. Emamectin is a soluble derivative of an avermectin. It is an insecticide, which
- PMID 27049309
- A pharmacological characterization of GABA, THIP and DS2 at binary α4β3 and β3δ receptors: GABA activates β3δ receptors via the β3(+)δ(-) interface.
- Lee H1, Absalom NL1, Hanrahan JR1, van Nieuwenhuijzen P1, Ahring PK1, Chebib M2.
- Brain research.Brain Res.2016 May 12. pii: S0006-8993(16)30373-0. doi: 10.1016/j.brainres.2016.05.019. [Epub ahead of print]
- There is growing evidence that GABA (γ-aminobutyric acid) can activate GABAA receptors (GABAARs) in the absence of an α subunit. In this study, we compared the pharmacology of homomeric and binary α4, β3 or δ subunits with ternary α4β3δ to identify subunit interfaces that contribute to the p
- PMID 27181518
Japanese Journal
- Isoxazoline insecticides : A novel class of GABA-gated chloride channel blockers(Molecular Targets for Insecticide Discovery II: GABA Receptors, Ion Channels, Acetylcholinesterases, Respiratory Chain…,1) Pest Management, Crop Protection and Vector Control)
- B219 イエバエ由来グルタミン酸依存性クロルイオンチャネル遺伝子及びGABA依存性クロルイオンチャネル遺伝子の発現解析
- Gunasekara Amrith S.,Truong Tresca,Goh Kean S. [他],SPURLOCK Frank,TJEERDEMA Ronald S.
- Journal of pesticide science = 日本農薬学会誌 32(3), 189-199, 2007-08-20
- … フィプロニルは比較的新しい殺虫剤で,広範な昆虫を低い投与濃度で制御する.その作用機作はγ-アミノ酪酸(GABA)依存性チャンネルの正常な機能を妨害することであり,数種類の昆虫に抵抗性が発達してきた有機りん剤やカーバメート剤のような古典的殺虫剤と対比させて,"新世代"殺虫剤と呼ばれている.フィプロニルは世界中で広く使用されており,毒性や環境運命についても多くの研究が行われている.本殺虫剤はある種の …
- NAID 110006379888
Related Links
- GABAは代表的抑制性神経伝達物質であり、中枢神経系のGABA-A受容体は、Benzodiazepine受容体、Picrotoxin結合部位、及びCl^-channelと複合体を形成し、Benzodiazepines、Barbiturates、及び、Bicuculline、Picrotoxinはこの ...
- 1870 Current Pharmaceutical Design, 2005, Vol. 11, No. 15 Graham A.R. Johnston extracellular N-terminus (α1, α2, α3 and α5 subunits). Mutation of this histidine to an arginine results in GABA A receptors that are insensitive to ...
Related Pictures
★リンクテーブル★
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- 関
- GABA-gated
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- 英
- GABAergic、GABA-gated
- 関
- GABA作働性
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- butyl
- 英
- γ-aminobutyric acid, γ-aminobutyrate, gamma aminobutyric acid
- 同
- γ-アミノ酪酸、4-アミノ酪酸、γ-アミノ酪酸、γアミノ酪酸、ガンマアミノブチル酸
- 関
- GABA受容体。ブチル
構造
生合成
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