- 関
- 5-HT agonist、5-HT1 agonist、5-HT2 agonist、serotonergic agonist、serotonin agonist、serotonin receptor agonist
WordNet
- (biochemistry) a drug that can combine with a receptor on a cell to produce a physiological reaction
- a muscle that contracts while another relaxes; "when bending the elbow the biceps are the agonist"
- someone involved in a contest or battle (as in an agon)
- the 8th letter of the Roman alphabet (同)h
PrepTutorEJDIC
- hydrogenの化学記号
- 鉛筆の硬度 / 《俗》heroin
UpToDate Contents
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English Journal
- The complex role of serotonin and 5-HT receptors in chronic pain.
- Bardin L.SourceDivision of Neurobiology 2, Centre de Recherche Pierre Fabre, Castres, France.
- Behavioural pharmacology.Behav Pharmacol.2011 Jul 29. [Epub ahead of print]
- Serotonin [5-hydroxytryptamine (5-HT)] in the central nervous system and in the periphery has long been considered to have an important role in the control of pain, for example, through descending inhibition. In recent years, considerable research efforts have focused on the role played by 5-HT on a
- PMID 21808193
- Discovery of 1-[2-(2,4-dimethylphenylsulfanyl)phenyl]piperazine (Lu AA21004): a novel multimodal compound for the treatment of major depressive disorder.
- Bang-Andersen B, Ruhland T, Jorgensen M, Smith G, Frederiksen K, Jensen KG, Zhong H, Nielsen SM, Hogg S, Mork A, Stensbol TB.SourceNeuroscience Drug Discovery Denmark, H. Lundbeck A/S , 9 Ottiliavej, DK-2500 Copenhagen-Valby, Denmark. ban@lundbeck.com
- Journal of medicinal chemistry.J Med Chem.2011 May 12;54(9):3206-21. Epub 2011 Apr 12.
- The synthesis and structure-activity relationship of a novel series of compounds with combined effects on 5-HT(3A) and 5-HT(1A) receptors and on the serotonin (5-HT) transporter (SERT) are described. Compound 5m (Lu AA21004) was the lead compound, displaying high affinity for recombinant human 5-HT(
- PMID 21486038
Japanese Journal
- Effects of Mosapride Citrate, a 5-HT4–Receptor Agonist, on Gastric Distension–Induced Visceromotor Response in Conscious Rats
- Seto Yasuhiro,Yoshida Naoyuki,Kaneko Hiroshi
- Journal of Pharmacological Sciences 116(1), 47-53, 2011
- … Mosapride citrate (mosapride), a prokinetic agent with 5-HT4–receptor agonistic activity, is known to enhance gastric emptying and alleviate symptoms in patients with functional dyspepsia (FD). … Additionally, a major metabolite M1 of mosapride, which possesses 5-HT3–receptor antagonistic activity, inhibited gastric distension–induced VMR. …
- NAID 130000663527
- Possible Involvement of β1 Receptors in Various Emetogen-Induced Increases in Salivary Amylase Activity in Rats
- Fukui Hideo,Suyama Yoshimi,Iwachido Takako,Miwa Eri
- Journal of Pharmacological Sciences advpub(0), 1012130486, 2010
- … We investigated the inhibitory effects of β1- or β2-adrenoceptor (AR) antagonists on salivary amylase secretion produced by various emetic agents, such as cisplatin, apomorphine, and lithium chloride (LiCl), or the non-emetic agent β1/2-AR agonist isoprenaline in rats. …
- NAID 130000439925
Related Links
- The 5-HT3 antagonists are a class of medications that act as receptor antagonists at the 5-HT3 receptor, a subtype of serotonin receptor found in terminals of the vagus nerve and in certain areas of the brain. With the notable exception ...
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- 関
- 5-HT1 agonist、5-HT2 agonist、5-HT3 agonist、serotonergic agent、serotonergic agonist、serotonin agonist、serotonin receptor agonist
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- 英
- 5-HT3 agonist
- 関
- セロトニン作動薬、5-HT1作動薬、セロトニン受容体作動薬、5-HT2作動薬、5-HT3アゴニスト、5-HT3作動薬、セロトニン刺激薬、セロトニン受容体刺激薬、5-HT3受容体刺激薬、5-HT2刺激薬
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- 英
- 5-HT3 agonist
- 関
- セロトニン作動薬、5-HT1作動薬、セロトニン受容体作動薬、5-HT2作動薬、5-HT3作動薬、セロトニン刺激薬、セロトニン受容体刺激薬、5-HT3刺激薬、5-HT3受容体刺激薬、5-HT2刺激薬
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- 関
- 5-HT agonist、5-HT1 agonist、5-HT2 agonist、5-HT3 agonist、serotonergic agent、serotonergic agonist、serotonin receptor agonist
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- 関
- 5-HT agonist、5-HT1 agonist、5-HT2 agonist、5-HT3 agonist、serotonergic agent、serotonin agonist、serotonin receptor agonist
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