- 関
- inhibitory activity、repression activity
WordNet
- the state of being potent; a males capacity to have sexual intercourse (同)potence
- capacity to produce strong physiological or chemical effects; "the toxins potency"; "the strength of the drinks" (同)effectiveness, strength
- a substance that retards or stops an activity
- restrictive of action; "a repressive regime"; "an overly strict and inhibiting discipline" (同)repressive, repressing
PrepTutorEJDIC
- 力,能力,権勢,影響力 / (薬などの)効能
- 抑制する人(物) / 化学反応抑制剤
UpToDate Contents
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English Journal
- Design, synthesis and biological evaluation of 4-benzoyl-1-dichlorobenzoylthiosemicarbazides as potent Gram-positive antibacterial agents.
- Paneth A1, Plech T1, Kaproń B1, Hagel D1, Kosikowska U2, Kuśmierz E1, Dzitko K3, Paneth P4.
- Journal of enzyme inhibition and medicinal chemistry.J Enzyme Inhib Med Chem.2016 Jun;31(3):434-40. doi: 10.3109/14756366.2015.1036050. Epub 2015 Apr 21.
- Twelve 4-benzoyl-1-dichlorobenzoylthiosemicarbazides have been tested as potential antibacterials. All the compounds had MICs between 0.49 and 15.63 µg/ml toward Micrococcus luteus, Bacillus cereus, Bacillus subtilis and Staphylococcus epidermidis indicating, in most cases, equipotent or even mor
- PMID 25897586
- Minocycline enhances inhibitory transmission to substantia gelatinosa neurons of the rat spinal dorsal horn.
- Peng HZ1, Ma LX1, Lv MH2, Hu T1, Liu T3.
- Neuroscience.Neuroscience.2016 Apr 5;319:183-93. doi: 10.1016/j.neuroscience.2016.01.047. Epub 2016 Jan 28.
- Minocycline, a second-generation tetracycline, is well known for its antibiotic, anti-inflammatory, and antinociceptive effects. Modulation of synaptic transmission is one of the analgesic mechanisms of minocycline. Although it has been reported that minocycline may suppress excitatory glutamatergic
- PMID 26826332
- Discovery of novel pyrrolo[2,3-b]pyridine derivatives bearing 1,2,3-triazole moiety as c-Met kinase inhibitors.
- Tang Q1, Wang L2, Tu Y2, Zhu W2, Luo R3, Tu Q2, Wang P2, Wu C2, Gong P4, Zheng P5.
- Bioorganic & medicinal chemistry letters.Bioorg Med Chem Lett.2016 Apr 1;26(7):1680-4. doi: 10.1016/j.bmcl.2016.02.059. Epub 2016 Feb 21.
- A series of novel pyrrolo[2,3-b]pyridine derivatives bearing 1,2,3-triazole moiety were designed, synthesized, and evaluated for their c-Met kinase inhibitory activities and antiproliferative activities against 4 cancer cell lines (HT-29, A549, MCF-7, and PC-3) in vitro. Most compounds showed modera
- PMID 26923692
Japanese Journal
- Synthesis of Clovamide Analogues That Inhibit NO Production in Activated BV-2 Microglial Cells
- Inhibitory Potency of Marketed Drugs for Ulcerative Colitis and Crohn's Disease on PEPT1
- Synthesis of Clovamide Analogues that Inhibit NO Production in Activated BV-2 Microglial Cells
Related Links
- In other words, it is the half maximal (50%) inhibitory concentration (IC) of a substance (50% IC, or IC50). It is commonly used as a measure of antagonist drug potency in pharmacological research. According to the FDA, IC50 represents the ...
- A medicinal enzyme inhibitor is often judged by its specificity (its lack of binding to other proteins) and its potency (its dissociation constant, which indicates the concentration needed to inhibit the enzyme). A high specificity and potency ensure ...
Related Pictures
★リンクテーブル★
[★]
- 英
- inhibitory activity、inhibitory potency、repression activity
- 関
- 阻害活性
[★]
- 関
- inhibitory potency、repression activity
[★]
- 英
- inhibitory activity、inhibitory potency
- 関
- 抑制活性
[★]
- 関
- inhibitory activity、inhibitory potency
[★]
- 関
- blocker、depressant、suppressant
[★]
- 関
- inhibiting、suppressive