Estrogenics
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Receptor
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ER (α, β)
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Agonists
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- 3α-Androstanediol
- 3β-Androstanediol
- 3α-Hydroxytibolone
- 3β-Hydroxytibolone
- 7-Oxo-DHEA
- 7α-Hydroxy-DHEA
- 7β-Hydroxyepiandrosterone
- 16α-Hydroxy-DHEA
- 16α-Hydroxyestrone
- Δ4-Androstenedione
- Δ5-Androstenediol
- 17α-Estradiol (alfatradiol)
- 17β-Estradiol (estradiol)
- Alestramustine
- Almestrone
- Benzestrol
- Bifluranol
- Broparestrol
- Carbestrol
- Chalconoids (e.g., isoliquiritigenin, phloretin, phlorizin (phloridzin), wedelolactone)
- Chlorotrianisene
- Cloxestradiol
- Conjugated equine estrogens (e.g., sodium equilin sulfate, sodium equilenin sulfate)
- Coumestans (e.g., coumestrol, psoralidin)
- DHEA
- DHEA-S
- Deoxymiroestrol
- Dienestrol
- Diethylstilbestrol
- Diethylstilbestrol diphosphate
- Diosgenin
- Doisynoestrol
- DPN
- DY-131 (GSK-9089)
- Epiestriol
- Epimestrol
- ERB-041
- Esterified estrogens (e.g., estrone sulfate, equilin sulfate, equilenin sulfate)
- Estetrol
- Estradiol benzoate
- Estradiol butyrylacetate
- Estradiol cypionate
- Estradiol dienanthate
- Estradiol dipropionate
- Estradiol diundecylate
- Estradiol diundecylenate
- Estradiol enanthate
- Estradiol furoate
- Estradiol hemihydrate
- Estradiol hemisuccinate
- Estradiol hexahydrobenzoate
- Estradiol monopropionate
- Estradiol palmitate
- Estradiol pivalate
- Estradiol propoxyphenylpropionate
- Estradiol stearate
- Estradiol succinate
- Estradiol undecylate
- Estradiol valerate
- Estramustine
- Estramustine phosphate
- Estrapronicate
- Estrazinol
- Estriol
- Estriol succinate
- Estriol tripropionate
- Estrofurate
- Estromustine
- Estrone
- Estrone acetate
- Estrone cyanate
- Estrone sulfate
- Estrone tetraacetylglucoside
- Estropipate
- Etamestrol (eptamestrol)
- Ethinyl estradiol
- Ethinyl estradiol 3-isopropylsulfonate
- Etynodiol diacetate
- FERb 033
- Fenestrel
- Flavonoids (incl. 7,8-DHF, 8-prenylnaringenin, apigenin, baicalein, baicalin, calycosin, catechin, daidzein, daidzin, ECG, EGCG, epicatechin, equol, formononetin, glabrene, glabridin, genistein, genistin, glycitein, kaempferol, liquiritigenin, mirificin, myricetin, naringenin, pinocembrin, prunetin, puerarin, quercetin, tectoridin, tectorigenin)
- Fosfestrol
- Furostilbestrol
- GSK-4716
- Hexestrol
- Hexestrol diacetate
- Hexestrol dicaprylate
- Hexestrol diphosphate
- Hexestrol dipropionate
- Hydroxyestrone diacetate
- Lignans (e.g., enterodiol, enterolactone)
- Mestranol
- Metalloestrogens (e.g., cadmium)
- Methallenestril
- Methestrol
- Methestrol dipropionate
- Miroestrol
- Moxestrol
- Nilestriol
- Orestrate
- Phytosterols (e.g., β-sitosterol, campesterol, stigmasterol)
- Polyestradiol phosphate
- PPT
- Promestriene
- Promethoestrol
- Resorcylic acid lactones (e.g., zearalanone, zearalenol, zearalenone, zeranal (zearalanol))
- Quinestradol
- Quinestrol
- Stilbenoids (e.g., resveratrol)
- Synthetic xenoestrogens (e.g., alkylphenols, bisphenols (e.g., BPA, BPF, BPS), DDT, parabens, PBBs, phthalates, PCBs)
- (R,R)-THC
- WAY-200070
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Mixed (SERMs)
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- 2-Hydroxyestrone
- 27-Hydroxycholesterol
- Acolbifene
- Afimoxifene
- Arzoxifene
- Bazedoxifene
- Clomifene
- Clomifenoxide
- Cyclofenil
- Droloxifene
- Enclomifene
- Endoxifen
- Epimestrol
- Femarelle
- Fispemifene
- GW5638
- Idoxifene
- Lasofoxifene
- Levormeloxifene
- Menerba
- Mepitiostane
- Miproxifene
- Nafoxidine
- Nitromifene
- Ormeloxifene
- Ospemifene
- Panomifene
- Pipendoxifene
- Prinaberel
- Raloxifene
- SS1010
- Sivifene
- Tamoxifen
- TAS-108
- Tesmilifene
- Tibolone
- Toremifene
- Trioxifene
- Y-134
- Zindoxifene
- Zuclomifene
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Antagonists
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- Fulvestrant
- ICI-164384
- MIBE
- MPP
- PHTPP
- RU-58668
- SS1020
- (R,R)-THC
- XCT-790
- ZK-164015
- ZK-191703
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GPER
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Agonists
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- 7β-Hydroxyepiandrosterone
- Afimoxifene
- Estradiol
- Fulvestrant
- G-1
- Genistein
- GPER-L1
- GPER-L2
- Niacin
- Nicotinamide
- PPT
- Quercetin
- Raloxifene
- Tamoxifen
- Tectoridin
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Antagonists
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Enzyme |
Modulators
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- See here instead (modulators of 20,22-desmolase, 17α-hydroxylase/17,20-lyase, 3β-HSD, 17β-HSD, 5α-reductase, aromatase, and 27-hydroxylase).
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Others |
Precursors
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- Cholesterol
- 22R-Hydroxycholesterol
- 20α,22R-Dihydroxycholesterol
- Pregnenolone
- Pregnenolone sulfate
- 17-Hydroxypregnenolone
- Progesterone
- 17-Hydroxyprogesterone
- 11-Deoxycortisol (cortodoxone)
- DHEA
- DHEA sulfate
- 16-Hydroxy-DHEA sulfate
- Δ5-Androstenediol
- Δ4-Androstenedione
- 16-Hydroxyandrostenedione
- Testosterone
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Indirect
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- Antigonadotropins (e.g., androgens, estrogens, progestogens, prolactin)
- Calcitriol (vitamin D)
- GnRH agonists (e,g, GnRH, leuprorelin)
- GnRH antagonists (e.g., cetrorelix)
- Gonadotropins (e.g., FSH, hCG, LH)
- Kisspeptin
- Plasma proteins (ABP, albumin, SHBG)
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See also: Androgenics • Glucocorticoids • Mineralocorticoids • Progestogenics
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