alpha-adrenergic antagonist

出典: meddic

alpha-adrenergic blocking agentalpha-adrenergic receptor antagonistalpha-blocker

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出典(authority):フリー百科事典『ウィキペディア(Wikipedia)』「2016/04/16 04:20:56」(JST)

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  • Investigation of the role of alpha-2 adrenergic receptors on prepulse inhibition of acoustic startle reflex in rats.
  • Ozcetin A1, Cevreli B1, Uzbay T2.
  • Synapse (New York, N.Y.).Synapse.2016 Dec;70(12):501-507. doi: 10.1002/syn.21923. Epub 2016 Jul 28.
  • OBJECTIVES: Alpha-2 adrenergic receptors target several behavioral functions. These receptors may connect with the brain pathways mediating sensorimotor gating system that associate with psychoses, and the literature that investigate the relationship between alpha-2 receptors and sensorimotor gating
  • PMID 27399264
  • Arylsulfonamide derivatives of (aryloxy)ethyl pyrrolidines and piperidines as α1-adrenergic receptor antagonist with uro-selective activity.
  • Rak A1, Canale V2, Marciniec K3, Żmudzki P2, Kotańska M1, Knutelska J1, Siwek A4, Stachowicz G4, Bednarski M5, Nowiński L6, Zygmunt M1, Zajdel P2, Sapa J1.
  • Bioorganic & medicinal chemistry.Bioorg Med Chem.2016 Nov 1;24(21):5582-5591. doi: 10.1016/j.bmc.2016.09.017. Epub 2016 Sep 10.
  • A series of arylsulfonamide derivatives of (aryloxy)ethyl pyrrolidines and piperidines was synthesized to develop new α1-adrenoceptor antagonists with uroselective profile. Biological evaluation for α1- and α2-adrenorecepor showed that tested compounds 13-37 displayed high-to-moderate affinity fo
  • PMID 27658792
  • Type-7 metabotropic glutamate receptors negatively regulate α1-adrenergic receptor signalling.
  • Iacovelli L1, Di Menna L2, Peterlik D3, Stangl C3, Orlando R1, Molinaro G2, De Blasi A4, Bruno V5, Battaglia G2, Flor PJ3, Uschold-Schmidt N3, Nicoletti F6.
  • Neuropharmacology.Neuropharmacology.2016 Oct 18. pii: S0028-3908(16)30468-3. doi: 10.1016/j.neuropharm.2016.10.018. [Epub ahead of print]
  • We studied the interaction between mGlu7 and α1-adrenergic receptors in heterologous expression systems, brain slices, and living animals. L-2-Amino-4-phosphonobutanoate (L-AP4), and l-serine-O-phosphate (L-SOP), which activate group III mGlu receptors, restrained the stimulation of polyphosphoinos
  • PMID 27769854


  • Natural course of lower urinary tract symptoms following discontinuation of alpha-1-adrenergic blockers in patients with benign prostatic hyperplasia
  • YOKOYAMA Teruhiko,WATANABE Toyohiko,SAIKA Takashi,NASU Yasutomo,KUMON Hiromi,MIYAJI Yoshiyuki,NAGAI Atsushi
  • International journal of urology 14(7), 598-601, 2007-07-01
  • … <p>alpha 1-adrenergic blockers (alpha b) remain the first-line therapy in men with lower urinary tract symptoms (LUTS). … The current published work advocates continued use of alpha b for their effect to be maintained. … In this study, we investigated the natural course of LUTS after the discontinuation of successful treatment of alpha b. …
  • NAID 10019725755
  • Effects of Ultrasonic Radiation on Cutaneous Blood Flow in the Paw of Decerebrated Rats
  • Nishimoto Chinami,Ishiura Yuichi,Kuniyasu Katsushi,Koga Tomoshige
  • Kawasaki journal of medical welfare 12(1), 13-18, 2006
  • … The increased blood flow continued even after the alpha-adrenergic receptor antagonist, phentolamine, was administered. …
  • NAID 120005358096
  • Effects of Ultrasonic Radiation on Cutaneous Blood Flow in the Paw of Decerebrated Rats
  • "Nishimoto Chinami,Ishiura Yuichi,Kuniyasu Katsushi,Koga Tomoshige"
  • Kawasaki journal of medical welfare 12(1), 13-18, 2006
  • … The increased blood flow continued even after the alpha-adrenergic receptor antagonist, phentolamine, was administered. …
  • NAID 110004745377


antagonist /an·tag·o·nist/ (an-tag´o-nist) 1. a substance that tends to nullify the action of another, as a drug that binds to a cell receptor without ... In addition, "emerging, exciting evidence" supports the use of the alpha-adrenergic ...
Alpha. Alpha measures risk-adjusted return, or the actual return an equity security provides in relation to the return you would expect based on its beta. Beta measures the security's volatility in relation to its benchmark index. If a ...



リンク元alpha-blocker」「αアドレナリン遮断薬」「alpha-adrenergic receptor antagonist」「αアドレナリン拮抗薬」「alpha-adrenergic blocking agent
関連記事alpha」「antagonist」「adrenergic」「adrenergic antagonist」「adrenergics



alpha-adrenergic antagonistalpha-adrenergic receptor antagonist



alpha-adrenergic antagonistalpha-adrenergic blocking agent

alpha-adrenergic receptor antagonist」


alpha-adrenergic antagonistalpha-blocker



alpha-adrenergic antagonist

alpha-adrenergic blocking agent」


alpha-adrenergic antagonist





WordNet   license wordnet

「first in order of importance; "the alpha male in the group of chimpanzees"; "the alpha star in a constellation is the brightest or main star"」

WordNet   license wordnet

「the 1st letter of the Greek alphabet」

WordNet   license wordnet

「the beginning of a series or sequence; "the Alpha and Omega, the first and the last, the beginning and the end"--Revelations」

PrepTutorEJDIC   license prepejdic

「アルファ(ギリシア語アルファベットの第1字A,α;英語のA,aに相当) / アルファ星(星座の主星)」

WordNet   license wordnet

「early testing stage of a software or hardware product; "alpha version"」


  [★] 拮抗薬

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「a drug that neutralizes or counteracts the effects of another drug」

WordNet   license wordnet

「a muscle that relaxes while another contracts; "when bending the elbow the triceps are the antagonist"」

PrepTutorEJDIC   license prepejdic




  • adj.
  • アドレナリンの、アドレナリン性の

WordNet   license wordnet

「drug that has the effects of epinephrine」
adrenergic drug

WordNet   license wordnet

「relating to epinephrine (its release or action)」

adrenergic antagonist」


adrenergic blockeradrenergic receptor antagonistadrenolyticsantiadrenergic agentantiadrenergics




adrenergicadrenergic agentadrenergic agonistadrenergic drugadrenergic receptor agonist