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1. 過敏性腸症候群に対するアロセトロン塩酸塩（Lotronex） alosetron hydrochloride lotronex for irritable bowel syndrome
2. 変形性関節症の初回薬物療法 initial pharmacologic therapy of osteoarthritis
3. クリンダマイシン：概要 clindamycin an overview
4. 成人における急性咽頭炎の対症療法 symptomatic treatment of acute pharyngitis in adults
5. 慢性非アレルギー性鼻炎 chronic nonallergic rhinitis

Determination of azasetron hydrochloride in rabbit plasma by liquid chromatography tandem mass spectrometry and its application.

Lin G1, Ma J, Zhu J, Yang X, Hu L, Wang X.
Biomedical chromatography : BMC.Biomed Chromatogr.2011 Oct;25(10):1107-11. doi: 10.1002/bmc.1578. Epub 2010 Dec 29.
A sensitive and selective liquid chromatography tandem mass spectrometry method for determination of azasetron hydrochloride in rabbit plasma was developed. After addition of doxapram hydrochloride as internal standard (IS), protein precipitation by 10% trichloroacetic acid was used as sample prepar
PMID 21204117

Study of 5HT3 and HT4 receptor expression in HT29 cell line and human colon adenocarcinoma tissues.

Ataee R1, Ajdary S, Rezayat M, Shokrgozar MA, Shahriari S, Zarrindast MR.
Archives of Iranian medicine.Arch Iran Med.2010 Mar;13(2):120-5.
BACKGROUND: Serotonin (5HT) has been shown to be a mitogenic factor in several carcinomas. Its mitogenic effect is elicited through a wide range of 5HT receptor subtypes. In this study, the effects of 5HT, 5HT3 (1-phenylbiguanide hydrochloride) and 5HT4 (cisapride) agonists in promoting the growth o
PMID 20187666

Y25130 hydrochloride, a selective 5HT3 receptor antagonist has potent antimitogenic and apoptotic effect on HT29 colorectal cancer cell line.

Ataee R1, Ajdary S, Zarrindast M, Rezayat M, Shokrgozar MA, Ataee A.
European journal of cancer prevention : the official journal of the European Cancer Prevention Organisation (ECP).Eur J Cancer Prev.2010 Mar;19(2):138-43. doi: 10.1097/CEJ.0b013e3283354901.
Serotonin (5-hydroxytryptamine, 5-HT) is known to be a mitogenic factor in several malignancies. It elicits its mitogenic effect through a wide range of 5-HT receptor subtypes and several internal cellular transcription pathways. According to wide distribution of 5-HT3 and 5-HT4 receptors in the gas
PMID 20010428

山田安彦,藤田美奈,奥山清 [他],高柳理早,大関健志,横山晴子,伊賀立二
藥學雜誌 127(2), 353-357, 2007-02-01
… We analyzed 5-HT_3 receptor occupancy of serotonin by integrating pharmacokinetic and receptor-binding kinetic parameters based on the receptor occupancy theory to compare the strength of the antiemetic effects of three dosage regimens of azasetron hydrochloride. …
NAID 110006163790

芳賀慶一郎,稲葉賢一,正路英典 [他],橋本敏夫
日本薬理学雑誌 116(5), 313-320, 2000-11-01
… The occurrence of delayed emesis induced 24 h after the administration of a non-platina chemotherapeutic agent, doxorubicin hydrochloride (doxorubicin), as well as behaviors such as feeding, drinking and defecation were examined in dogs. … azasetron, a 5-HT<SUB>3</SUB> … Azasetron was found to improve the increased frequency of defecation, but exerted no obvious effect on hypophagia or on the decreased frequency of drinking. …
NAID 10008181341