vasopressin receptor agonist

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  • Vasopressin V1a and V1b receptor modulators: a patent review (2012 - 2014).
  • Ślusarz MJ1.
  • Expert opinion on therapeutic patents.Expert Opin Ther Pat.2015 Jun;25(6):711-22. doi: 10.1517/13543776.2015.1026257. Epub 2015 Mar 16.
  • INTRODUCTION: The vasopressin V1a and V1b receptors are involved in many crucial physiological, reproductive, behavioral and social functions. Consequently, they are also involved in several pathological conditions, thus the ligands capable of selective stimulation/inhibition of these receptors may
  • PMID 25776143
  • The novel desmopressin analogue [V4Q5]dDAVP inhibits angiogenesis, tumour growth and metastases in vasopressin type 2 receptor-expressing breast cancer models.
  • Garona J1, Pifano M1, Orlando UD2, Pastrian MB3, Iannucci NB3, Ortega HH4, Podesta EJ2, Gomez DE1, Ripoll GV1, Alonso DF1.
  • International journal of oncology.Int J Oncol.2015 Jun;46(6):2335-45. doi: 10.3892/ijo.2015.2952. Epub 2015 Apr 3.
  • Desmopressin (dDAVP) is a safe haemostatic agent with previously reported antitumour activity. It acts as a selective agonist for the V2 vasopressin membrane receptor (V2r) present on tumour cells and microvasculature. The purpose of this study was to evaluate the novel peptide derivative [V4Q5]dDA
  • PMID 25846632


  • The efficacy and safety of terlipressin and albumin in patients with type 1 hepatorenal syndrome : a multicenter, open-label, explorative study
  • Oxytocin and dopamine stimulate ghrelin secretion by the ghrelin-producing cell line, MGN3-1 in vitro.
  • Changes in vasopressin release and autonomic function induced by manipulating forebrain GABAergic signaling under euvolemia and hypovolemia in conscious rats


1. Br J Pharmacol. 2013 Sep;170(2):278-92. doi: 10.1111/bph.12249. Pharmacological characterization of FE 201874, the first selective high affinity rat V1A vasopressin receptor agonist. Marir R, Virsolvy A, Wisniewski K, Mion J ...
Calcium antagonizes the magnesium-induced high affinity state of the hepatic vasopressin receptor for the agonist interaction. Your browsing activity is empty. Activity recording is turned off. Turn recording back on Links Compound ...



関連記事agonist」「vasopressin」「receptor」「receptor agonist」「vasopressin receptor


  [★] 作動薬

WordNet   license wordnet

「(biochemistry) a drug that can combine with a receptor on a cell to produce a physiological reaction」

WordNet   license wordnet

「a muscle that contracts while another relaxes; "when bending the elbow the biceps are the agonist"」

WordNet   license wordnet

「someone involved in a contest or battle (as in an agon)」


  [★] バソプレシン

WordNet   license wordnet

「hormone secreted by the posterior pituitary gland (trade name Pitressin) and also by nerve endings in the hypothalamus; affects blood pressure by stimulating capillary muscles and reduces urine flow by affecting reabsorption of water by kidney tubules」
antidiuretic hormone, ADH, Pitressin


  [★] 受容体

WordNet   license wordnet

「a cellular structure that is postulated to exist in order to mediate between a chemical agent that acts on nervous tissue and the physiological response」

PrepTutorEJDIC   license prepejdic

「=sense organ / 受信装置」

receptor agonist」



vasopressin receptor」

  [★] バソプレシン受容体